Protein inhibitor inhengo inobatanidza kune catalyst, ichitadzisa kuita kwayo. Catalysts, ari mapuroteni anobatsira mhinduro dzemukomboni nekusingaperi, anoshanda neshanduko ye substrate particles kuita zvigadzirwa.[1] Mushonga unozadzisa izvi nekudzora substrate kunzvimbo yayo ine simba, imwe nzvimbo inomhanyisa danho rakaoma kwazvo remhinduro.


Protein inhibitor inopindirana mukutenderera uku neimwe kana imwe ichingomira kune kemikari ine simba saiti, ichichengeta substrate kubva pakudzora, kana kudzora kune imwezve saiti pakomboni, zvichiodza mwoyo catalyst's catalysis yemhinduro. Inhibitors inogona kuratidza kudzoreredza kana kusadzoreka. Irreversible inhibitors inogadzira chisungo chemusanganiswa neprotein, ichiidzvinyirira kusvikira chisungo chaputsika. 


Neimwe nzira, reversible inhibitors inosunga isina-covalently uye inogona kubva yazvitsaura kubva kune inokonzeresa, ichibvumira puroteni kuti ienderere mberi nekugona kwayo. Zvichienderana nekuti vanobatana here nekemikari, iyo compound substrate complex, kana zvese, reversible inhibitors zvinokonzeresa marudzi akasiyana ekuzvidzora.


Inhibitors

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  • Vismodegib

    CAS Kwete: 879085-55-9
    Chitarisiko: Kubva chena kana Yero hupfu kana Crystal
    Standard: mumba
    Kushandisa: Anti bundu; anti-cancer 
    Kugovera Mano: 50kg pamwedzi
    Kuchena: ≥99%
    Kubhadhara: T/T, LC kana DA
    Nguva Yekutumira: Yakagadzirira Stock muNharaunda Warehouse, 1-3 mazuva
    Origin: China
    Kutumira: DHL, FedEx, TNT, EMS, NeGungwa, Nemhepo
    Haikwanisi kutengesera vanhu
  • Purogiramu inonzi Verteporfin

    CAS Kwete: 129497-78-5
    Chitarisiko: Yakasvibira yakasvibira kusvika kutema yakasimba
    Standard: mumba
    Kushanda: Tsvakurudzo yeLab 
    Kugovera Mano: 100g pamwedzi
    Kuchena: ≥96%
    Kubhadhara: T/T, LC kana DA
    Nguva Yekutumira: Yakagadzirira Stock muNharaunda Warehouse, 1-3 mazuva
    Origin: China
    Kutumira: DHL, FedEx, TNT, EMS, NeGungwa, Nemhepo
    Haikwanisi kutengesera vanhu
  • EPZ-6438

    CAS Kwete: 1403254-99-8
    Kuonekwa: Ichena kana isina-white crystalline powder
    Standard: mumba
    Kushanda: Tsvakurudzo yeLab  
    Kugovera Mano: 1000g pamwedzi
    Kuchena: ≥98%
    Kubhadhara: T/T, LC kana DA
    Nguva Yekutumira: Yakagadzirira Stock muNharaunda Warehouse, 1-3 mazuva
    Origin: China
    Kutumira: DHL, FedEx, TNT, EMS, NeGungwa, Nemhepo
    Haikwanisi kutengesera vanhu
  • Alagebrium Chloride

    CAS Kwete: 341028-37-3
    Kuonekwa: inenge chena kana chena ruvara rwehupfu
    Standard: mumba
    Kugovera Mano: 1000g pamwedzi
    Kuchena: ≥99%
    Kubhadhara: T/T, LC kana DA
    Nguva Yekutumira: Yakagadzirira Stock muNharaunda Warehouse, 1-3 mazuva
    Origin: China
    Kutumira: DHL, FedEx, TNT, EMS, NeGungwa, Nemhepo
    Haikwanisi kutengesera vanhu
  • AZD 1480

    CAS Kwete: 935666-88-9
    Kuonekwa: kuchena kune beige powder
    Standard: mumba
    Kugovera Mano: 1000g pamwedzi
    Kuchena: ≥99%
    Kubhadhara: T/T, LC kana DA
    Nguva Yekutumira: Yakagadzirira Stock muNharaunda Warehouse, 1-3 mazuva
    Origin: China
    Kutumira: DHL, FedEx, TNT, EMS, NeGungwa, Nemhepo
    Haikwanisi kutengesera vanhu
  • AZD 8055

    CAS Kwete: 1009298-09-2
    Kutaridzika
    Standard: mumba
    Kugovera Mano: 1000g pamwedzi
    Kuchena: ≥99%
    Kubhadhara: T/T, LC kana DA
    Nguva Yekutumira: Yakagadzirira Stock muNharaunda Warehouse, 1-3 mazuva
    Origin: China
    Kutumira: DHL, FedEx, TNT, EMS, NeGungwa, Nemhepo
    Haikwanisi kutengesera vanhu
  • Clascoterone poda

    CAS Kwete: 19608-29-8
    Kuonekwa: kuchena kune chiedza chepfu yero
    Standard: mumba
    Kugovera Mano: 100kg pamwedzi
    Kuchena: ≥99%
    Kubhadhara: T/T, LC kana DA
    Nguva Yekutumira: Yakagadzirira Stock muNharaunda Warehouse, 1-3 mazuva
    Origin: China
    Kutumira: DHL, FedEx, TNT, EMS, NeGungwa, Nemhepo
    Haikwanisi kutengesera vanhu
  • Setipiprant powder

    CAS Kwete: 866460-33-5
    Kuonekwa: light yellow powder
    Standard: mumba
    Kugovera Mano: 1000g pamwedzi
    Kuchena: ≥99%
    Kubhadhara: T/T, LC kana DA
    Nguva Yekutumira: Yakagadzirira Stock muNharaunda Warehouse, 1-3 mazuva
    Origin: China
    Kutumira: DHL, FedEx, TNT, EMS, NeGungwa, Nemhepo
    Haikwanisi kutengesera vanhu
  • Pyrilutamide

    CAS Kwete: 1272719-00-2
    Kuonekwa: kuchena kune chiedza chepfu yero
    Standard: mumba
    Kugovera Mano: 1000g pamwedzi
    Kuchena: ≥99%
    Kubhadhara: T/T, LC kana DA
    Nguva Yekutumira: Yakagadzirira Stock muNharaunda Warehouse, 1-3 mazuva
    Origin: China
    Kutumira: DHL, FedEx, TNT, EMS, NeGungwa, Nemhepo
    Haikwanisi kutengesera vanhu
  • Purogiramu inonzi Finerenone

    CAS Kwete: 1050477-31-0
    Chitarisiko: Ichena kune yero crystalline poda
    Standard: mumba
    Kugovera Mano: 5000g pamwedzi
    Kuchena: ≥99%
    Kubhadhara: T/T, LC kana DA
    Nguva Yekutumira: Yakagadzirira Stock muNharaunda Warehouse, 1-3 mazuva
    Origin: China
    Kutumira: DHL, FedEx, TNT, EMS, NeGungwa, Nemhepo
    Haikwanisi kutengesera vanhu
  • Glecaprevir

    CAS: 1365970-03-1
    Chitarisiko: Muchena kune Off-White poda
    Kuchengeta: 98%
    Mucherechedzo: YIHUI
    Kutakura: 1g; 10g; 100g
    Kugovera Mano: 2000g pamwedziSherufu Hupenyu: Makore maviri
    Chikumbiro: Lab research
    Kubhadhara: T/T, LC kana DA
    Muenzaniso: iripo
    Nguva Yekutumira: Yakagadzirira Stock muNharaunda Warehouse, mazuva 1-3
    Kurumidza uye Kuchengetedza Kutumira
    Origin: China
    Kutumira: DHL, FedEx, TNT, EMS,Negungwa,Nemhepo
    Certifications: ISO9001, ISO22000, HACCP, HALAL, KOSHER
    Haikwanisi kutengesera vanhu
  • RTA-408

    CAS: 1474034-05-3
    Kuonekwa: Off- chena poda
    Kuchengeta: 98%
    Mucherechedzo: YIHUI
    Kutakura: 1g; 10g; 100g
    Kugovera Mano: 2000g pamwedzi
    Sherufu Hupenyu: Makore maviri
    Chikumbiro: Lab research
    Kubhadhara: T/T, LC kana DA
    Muenzaniso: iripo
    Nguva Yekutumira: Yakagadzirira Stock muNharaunda Warehouse, mazuva 1-3
    Kurumidza uye Kuchengetedza Kutumira
    Origin: China
    Kutumira: DHL, FedEx, TNT, EMS,Negungwa,Nemhepo
    Certifications: ISO9001, ISO22000, HACCP, HALAL, KOSHER
    Haikwanisi kutengesera vanhu
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